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Crizotinib

Synonyms

SourcesNames Used
CCLE, GRAYPF-2341066
GDSC1000, FIMMCrizotinib
gCSI, CTRPv2crizotinib
PharmacoGx Crizotinib

External IDs

DatabaseIdentifier
Smiles: CC(C1=C(C=C(C=C1Cl)F)Cl)OC2=C(N=CC(=C2)C3=CN(N=C3)C4CCNCC4)N
Inchikey: SCJHEFQWKWHQTO-GFCCVEGCSA-N
Pubchem: 54613769

Annotated Targets

MET, ALK

FDA Approval Status

Approved
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Top molecular features associated with response to Crizotinib


Feature TypeStandardized
Nominal ANOVA
mRNA NKG7 GDSC1000 pan-cancer AAC 0.32 8e-09
mRNA CLDN22 GDSC1000 pan-cancer AAC 0.29 1e-08
mRNA SWAP70 GDSC1000 pan-cancer AAC -0.3 1e-08
mRNA DMBX1 CTRPv2 pan-cancer AAC 0.18 2e-08
mRNA CAPZA2 gCSI pan-cancer AAC 0.33 2e-08
mRNA SEC31B CTRPv2 pan-cancer AAC 0.18 2e-08
mRNA OSM GDSC1000 pan-cancer AAC 0.32 2e-08
mRNA ANK1 CTRPv2 pan-cancer AAC 0.18 2e-08
mRNA CLEC4F GDSC1000 pan-cancer AAC 0.28 2e-08
mRNA CTSB GDSC1000 pan-cancer AAC 0.35 2e-08
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