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Crizotinib

Synonyms

SourcesNames Used
CCLE, GRAYPF-2341066
GDSC1000, FIMMCrizotinib
gCSI, CTRPv2crizotinib
PharmacoGx Crizotinib

External IDs

DatabaseIdentifier
Smiles: CC(C1=C(C=C(C=C1Cl)F)Cl)OC2=C(N=CC(=C2)C3=CN(N=C3)C4CCNCC4)N
Inchikey: SCJHEFQWKWHQTO-GFCCVEGCSA-N
Pubchem: 54613769

Annotated Targets

MET, ALK

FDA Approval Status

Approved
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Top molecular features associated with response to Crizotinib


Feature TypeStandardized
Nominal ANOVA
mRNA FAM46C GDSC1000 pan-cancer AAC 0.17 0.003
mRNA AP1B1 gCSI pan-cancer AAC -0.16 0.003
mRNA ANKMY2 CCLE pan-cancer AAC 0.14 0.003
mRNA TMEM133 CCLE pan-cancer AAC -0.14 0.003
mRNA FAM46C CCLE pan-cancer AAC 0.15 0.003
mRNA SPATA9 CTRPv2 pan-cancer AAC 0.095 0.003
mRNA SNX22 CCLE pan-cancer AAC -0.15 0.003
mRNA SUPT7L CTRPv2 pan-cancer AAC 0.098 0.003
mRNA MTNR1A CTRPv2 pan-cancer AAC 0.095 0.003
mRNA SIGLEC8 CTRPv2 pan-cancer AAC 0.096 0.003
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