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Crizotinib

Synonyms

SourcesNames Used
CCLE, GRAYPF-2341066
GDSC1000, FIMMCrizotinib
gCSI, CTRPv2crizotinib
PharmacoGx Crizotinib

External IDs

DatabaseIdentifier
Smiles: CC(C1=C(C=C(C=C1Cl)F)Cl)OC2=C(N=CC(=C2)C3=CN(N=C3)C4CCNCC4)N
Inchikey: SCJHEFQWKWHQTO-GFCCVEGCSA-N
Pubchem: 54613769

Annotated Targets

MET, ALK

FDA Approval Status

Approved
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Top molecular features associated with response to Crizotinib


Feature TypeStandardized
Nominal ANOVA
mRNA NPY5R FIMM pan-cancer AAC 0.49 0.003
mRNA ARL15 FIMM pan-cancer AAC 0.49 0.002
mRNA ZNF510 FIMM pan-cancer AAC 0.5 0.003
mRNA ATRNL1 FIMM pan-cancer AAC 0.5 0.002
mRNA MOSPD2 FIMM pan-cancer AAC 0.5 0.003
mRNA INPP4B FIMM pan-cancer AAC 0.51 0.002
mRNA JAK2 FIMM pan-cancer AAC 0.52 0.003
mRNA PGM5 FIMM pan-cancer AAC 0.52 0.001
mRNA SLC19A2 FIMM pan-cancer AAC 0.52 0.002
mRNA PARD6B FIMM pan-cancer AAC 0.53 0.001
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