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Crizotinib

Synonyms

SourcesNames Used
CCLE, GRAYPF-2341066
GDSC1000, FIMMCrizotinib
gCSI, CTRPv2crizotinib
PharmacoGx Crizotinib

External IDs

DatabaseIdentifier
Smiles: CC(C1=C(C=C(C=C1Cl)F)Cl)OC2=C(N=CC(=C2)C3=CN(N=C3)C4CCNCC4)N
Inchikey: SCJHEFQWKWHQTO-GFCCVEGCSA-N
Pubchem: 54613769

Annotated Targets

MET, ALK

FDA Approval Status

Approved
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Top molecular features associated with response to Crizotinib


Feature TypeStandardized
Nominal ANOVA
mRNA COQ8A CTRPv2 pan-cancer AAC 0.19 1e-07
mRNA NCR1 GDSC1000 pan-cancer AAC 0.27 1e-07
mRNA SWAP70 CTRPv2 pan-cancer AAC -0.17 1e-07
mRNA ROR2 GDSC1000 pan-cancer AAC 0.28 2e-07
mRNA USP32 GDSC1000 pan-cancer AAC 0.27 2e-07
mRNA RBM44 GDSC1000 pan-cancer AAC 0.26 2e-07
mRNA MLXIPL CTRPv2 pan-cancer AAC 0.18 2e-07
mRNA EAF2 GDSC1000 pan-cancer AAC -0.4 2e-07
mRNA ARHGAP15 CTRPv2 pan-cancer AAC 0.21 3e-07
mRNA IL1RAP GDSC1000 pan-cancer AAC 0.31 3e-07
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