| Erlotinib | CCLE, GDSC1000, gCSI, GRAY, FIMM, CTRPv2, UHNBreast | 2345 |
| lapatinib | CCLE, GDSC1000, gCSI, GRAY, FIMM, CTRPv2, UHNBreast | 2302 |
| Gefitinib | GDSC1000, GRAY, FIMM, CTRPv2 | 1948 |
| Vandetanib | CCLE, FIMM, CTRPv2 | 1381 |
| CUDC-101 | GDSC1000 | 975 |
| Cetuximab | GDSC1000 | 912 |
| neratinib | CTRPv2 | 867 |
| canertinib | CTRPv2 | 818 |
| WZ8040 | CTRPv2 | 754 |
| PD 153035 | CTRPv2 | 624 |