| GDC-0941 | GDSC1000, gCSI, FIMM, CTRPv2 | 3124 |
| AZD6482 | GDSC1000, CTRPv2 | 2756 |
| PI-103 | GDSC1000, CTRPv2 | 1835 |
| ZSTK474 | GDSC1000, CTRPv2 | 1826 |
| NVP-BEZ235 | GDSC1000, GRAY, CTRPv2 | 1597 |
| TGX221 | GDSC1000, CTRPv2 | 1287 |
| GSK2126458 | GDSC1000, GRAY | 1065 |
| TG-100-115 | CTRPv2 | 855 |
| XL765 | CTRPv2 | 834 |
| rigosertib | CTRPv2 | 823 |