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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA LBR CTRPv2 pan-cancer AAC 0.24 2e-08
mRNA DOT1L CTRPv2 pan-cancer AAC 0.26 2e-08
mRNA MYO1F GDSC1000 pan-cancer AAC 0.22 2e-08
mRNA FAM212A GDSC1000 pan-cancer AAC 0.21 2e-08
mRNA NFATC3 CTRPv2 pan-cancer AAC 0.26 2e-08
mRNA SFPQ CTRPv2 pan-cancer AAC 0.21 3e-08
mRNA GBGT1 GDSC1000 pan-cancer AAC 0.19 3e-08
mRNA ZYX GDSC1000 pan-cancer AAC 0.2 3e-08
mRNA RNASE3 GDSC1000 pan-cancer AAC 0.19 4e-08
mRNA CPSF6 CTRPv2 pan-cancer AAC 0.22 4e-08
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