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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA LMO2 GDSC1000 pan-cancer AAC 0.22 6e-09
mRNA RAB37 GDSC1000 pan-cancer AAC 0.23 7e-09
mRNA NIPAL3 CTRPv2 pan-cancer AAC -0.22 7e-09
mRNA ANXA5 CTRPv2 pan-cancer AAC -0.28 7e-09
mRNA BRD3 CTRPv2 pan-cancer AAC 0.22 7e-09
mRNA FAM78A GDSC1000 pan-cancer AAC 0.27 8e-09
mRNA ARHGAP19-SLIT1 CTRPv2 pan-cancer AAC 0.25 9e-09
mRNA ADGRE2 GDSC1000 pan-cancer AAC 0.21 1e-08
mRNA PTPN7 GDSC1000 pan-cancer AAC 0.32 1e-08
mRNA LILRB2 GDSC1000 pan-cancer AAC 0.2 1e-08
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