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OSI-930

Synonyms

SourcesNames Used
GDSC1000, CTRPv2OSI-930
PharmacoGx OSI-930

External IDs

DatabaseIdentifier
Smiles: FC(F)(F)Oc1ccc(NC(=O)c2sccc2NCc2ccnc3ccccc23)cc1
Pubchem: 9868037

Annotated Targets

KIT, KDR, FLT1

FDA Approval Status

Not Approved
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Top molecular features associated with response to OSI-930


Feature TypeStandardized
Nominal ANOVA
mRNA GHRL GDSC1000 pan-cancer AAC 0.21 6e-10
mRNA AIF1 GDSC1000 pan-cancer AAC 0.25 9e-10
mRNA LILRA1 GDSC1000 pan-cancer AAC 0.21 9e-10
mRNA TYROBP GDSC1000 pan-cancer AAC 0.22 1e-09
mRNA ZNF711 CTRPv2 pan-cancer AAC 0.24 2e-09
mRNA CLEC5A GDSC1000 pan-cancer AAC 0.2 3e-09
mRNA HCFC1 CTRPv2 pan-cancer AAC 0.24 3e-09
mRNA CD33 GDSC1000 pan-cancer AAC 0.22 4e-09
mRNA CYSLTR1 GDSC1000 pan-cancer AAC 0.23 4e-09
mRNA HNRNPU CTRPv2 pan-cancer AAC 0.22 5e-09
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