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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA TC2N CCLE pan-cancer AAC 0.34 3e-10
mRNA PKP3 CTRPv2 pan-cancer AAC 0.29 3e-10
mRNA FRK CCLE pan-cancer AAC 0.32 3e-10
mRNA TMC4 CCLE pan-cancer AAC 0.35 3e-10
mRNA PPL CCLE pan-cancer AAC 0.38 4e-10
mRNA SH2D3A gCSI pan-cancer AAC 0.39 4e-10
mRNA MST1R CCLE pan-cancer AAC 0.36 4e-10
mRNA CYP4F11 GDSC1000 pan-cancer AAC 0.35 4e-10
mRNA F3 gCSI pan-cancer AAC 0.41 4e-10
mRNA VGLL1 gCSI pan-cancer AAC 0.37 4e-10
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