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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA MARVELD2 CCLE pan-cancer AAC 0.4 1e-10
mRNA ESRP2 CCLE pan-cancer AAC 0.39 1e-10
mRNA BTC CCLE pan-cancer AAC 0.32 1e-10
mRNA CXCL16 CCLE pan-cancer AAC 0.34 1e-10
mRNA LCN2 CCLE pan-cancer AAC 0.34 2e-10
mRNA LAMA3 gCSI pan-cancer AAC 0.42 2e-10
mRNA KRT6A CCLE pan-cancer AAC 0.31 2e-10
mRNA JUP CCLE pan-cancer AAC 0.34 2e-10
mRNA GJB3 CTRPv2 pan-cancer AAC 0.27 2e-10
mRNA IRF6 CTRPv2 pan-cancer AAC 0.28 2e-10
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