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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA ELMO3 CCLE pan-cancer AAC 0.35 5e-11
mRNA LAD1 CCLE pan-cancer AAC 0.35 5e-11
mRNA CDH3 gCSI pan-cancer AAC 0.43 7e-11
mRNA ZEB1 CCLE pan-cancer AAC -0.32 8e-11
mRNA EPHA1 CCLE pan-cancer AAC 0.33 8e-11
mRNA FAM83H CCLE pan-cancer AAC 0.38 9e-11
mRNA ESRP1 CCLE pan-cancer AAC 0.35 9e-11
mRNA TNK1 CCLE pan-cancer AAC 0.35 9e-11
mRNA LAMC2 CCLE pan-cancer AAC 0.34 1e-10
mRNA GJB5 CCLE pan-cancer AAC 0.35 1e-10
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