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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA TMEM158 CCLE pan-cancer AAC -0.24 4e-06
mRNA C16orf45 CCLE pan-cancer AAC -0.24 6e-06
mRNA SYT4 gCSI pan-cancer AAC -0.24 0.0001
mRNA TTL CCLE pan-cancer AAC -0.24 2e-06
mRNA ZNF333 gCSI pan-cancer AAC -0.24 0.0001
mRNA SLC25A33 gCSI pan-cancer AAC -0.24 5e-05
mRNA CHST1 gCSI pan-cancer AAC -0.24 7e-05
mRNA C12orf57 gCSI pan-cancer AAC -0.24 2e-05
mRNA CNPY4 gCSI pan-cancer AAC -0.24 0.0001
mRNA EIF1B gCSI pan-cancer AAC -0.24 0.0001
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