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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA SCG2 gCSI pan-cancer AAC -0.26 2e-05
mRNA SPARC CCLE pan-cancer AAC -0.26 2e-05
mRNA AP4M1 gCSI pan-cancer AAC -0.26 3e-06
mRNA P3H1 CCLE pan-cancer AAC -0.26 1e-06
mRNA FMC1 gCSI pan-cancer AAC -0.26 6e-06
mRNA LRRC49 CCLE pan-cancer AAC -0.26 3e-06
mRNA PTMS gCSI pan-cancer AAC -0.25 0.0004
mRNA SYDE1 CCLE pan-cancer AAC -0.25 3e-06
mRNA ZNF775 gCSI pan-cancer AAC -0.25 4e-05
mRNA AP1S2 CCLE pan-cancer AAC -0.25 8e-06
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