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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA AP1M1 CCLE pan-cancer AAC -0.29 1e-08
mRNA ELAVL4 gCSI pan-cancer AAC -0.28 0.0001
mRNA SLC43A1 gCSI pan-cancer AAC -0.28 0.0002
mRNA DPYSL3 GDSC1000 pan-cancer AAC -0.28 1e-05
mRNA NXPE3 CCLE pan-cancer AAC -0.28 5e-08
mRNA PTPRN2 gCSI pan-cancer AAC -0.27 1e-06
mRNA LEF1 gCSI pan-cancer AAC -0.27 4e-05
mRNA CCDC88A CCLE pan-cancer AAC -0.26 2e-07
mRNA ST3GAL2 CCLE pan-cancer AAC -0.26 2e-07
mRNA PXK CCLE pan-cancer AAC -0.26 2e-06
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