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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA ZEB1 CCLE pan-cancer AAC -0.32 8e-11
mRNA ZEB1 CTRPv2 pan-cancer AAC -0.15 3e-05
mRNA ZEB2 CCLE pan-cancer AAC -0.22 0.0001
mRNA ZFP36 GDSC1000 pan-cancer AAC 0.28 3e-06
mRNA ZFYVE21 CCLE pan-cancer AAC 0.23 2e-05
mRNA ZFYVE21 CTRPv2 pan-cancer AAC 0.14 0.0003
mRNA ZHX3 CTRPv2 pan-cancer AAC -0.15 0.0001
mRNA ZKSCAN3 gCSI pan-cancer AAC -0.23 6e-05
mRNA ZKSCAN5 gCSI pan-cancer AAC -0.21 0.0002
mRNA ZMAT5 gCSI pan-cancer AAC -0.21 0.0001
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