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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA CHST10 CCLE pan-cancer AAC -0.18 0.0003
mRNA B3GALT4 CCLE pan-cancer AAC 0.18 0.0003
mRNA HRASLS5 gCSI pan-cancer AAC 0.2 0.0003
mRNA WHAMM GDSC1000 pan-cancer AAC 0.2 0.0003
mRNA GABRP gCSI pan-cancer AAC 0.2 0.0003
mRNA DPP4 FIMM pan-cancer AAC 0.63 0.0003
mRNA SMIM5 CCLE pan-cancer AAC 0.17 0.0003
mRNA NRBF2 FIMM pan-cancer AAC -0.7 0.0003
mRNA TMBIM1 gCSI pan-cancer AAC 0.23 0.0003
mRNA HTATSF1 GDSC1000 pan-cancer AAC -0.19 0.0003
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