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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA MMP7 gCSI pan-cancer AAC 0.22 0.0002
mRNA CARD6 CTRPv2 pan-cancer AAC 0.13 0.0002
mRNA MUS81 CTRPv2 pan-cancer AAC -0.13 0.0002
mRNA WFDC5 GDSC1000 pan-cancer AAC 0.18 0.0002
mRNA SAA2 gCSI pan-cancer AAC 0.21 0.0002
mRNA NRIP1 gCSI pan-cancer AAC 0.23 0.0002
mRNA ANO1 CCLE pan-cancer AAC 0.2 0.0002
mRNA MYZAP UHNBreast pan-cancer AAC 0.83 0.0002
mRNA BUD31 gCSI pan-cancer AAC -0.2 0.0002
mRNA THRB gCSI pan-cancer AAC 0.26 0.0002
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