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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA TSPAN1 CCLE pan-cancer AAC 0.35 5e-10
mRNA F11R CCLE pan-cancer AAC 0.34 5e-10
mRNA CAPN1 CCLE pan-cancer AAC 0.32 6e-10
mRNA CRB3 CCLE pan-cancer AAC 0.34 6e-10
mRNA SCEL CCLE pan-cancer AAC 0.32 6e-10
mRNA RHOD CCLE pan-cancer AAC 0.36 7e-10
mRNA RARRES3 gCSI pan-cancer AAC 0.35 7e-10
mRNA CEACAM6 CTRPv2 pan-cancer AAC 0.21 7e-10
mRNA ZNF165 CCLE pan-cancer AAC 0.34 8e-10
mRNA GPR87 gCSI pan-cancer AAC 0.4 8e-10
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