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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA ERP27 CCLE pan-cancer AAC 0.27 1e-08
mRNA RASEF CCLE pan-cancer AAC 0.29 1e-08
mRNA SCEL gCSI pan-cancer AAC 0.36 1e-08
mRNA CORO2A CCLE pan-cancer AAC 0.27 1e-08
mRNA NIPAL1 CCLE pan-cancer AAC 0.31 1e-08
mRNA FAM83B gCSI pan-cancer AAC 0.41 1e-08
mRNA GALNT3 CTRPv2 pan-cancer AAC 0.22 1e-08
mRNA KCNJ13 FIMM pan-cancer AAC 0.77 2e-08
mRNA BICDL2 CCLE pan-cancer AAC 0.32 2e-08
mRNA NTN4 gCSI pan-cancer AAC 0.38 2e-08
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