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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA SSH3 CCLE pan-cancer AAC 0.33 7e-09
mRNA TTC22 CTRPv2 pan-cancer AAC 0.22 7e-09
mRNA LPAR2 CCLE pan-cancer AAC 0.3 8e-09
mRNA TMEM265 CTRPv2 pan-cancer AAC 0.22 9e-09
mRNA GRHL1 CCLE pan-cancer AAC 0.3 9e-09
mRNA SOX15 CCLE pan-cancer AAC 0.29 1e-08
mRNA CST6 gCSI pan-cancer AAC 0.33 1e-08
mRNA PTGES gCSI pan-cancer AAC 0.37 1e-08
mRNA AP1M1 CCLE pan-cancer AAC -0.29 1e-08
mRNA TMPRSS11E CTRPv2 pan-cancer AAC 0.2 1e-08
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