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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA CDS1 CTRPv2 pan-cancer AAC 0.24 4e-09
mRNA KCNK1 CCLE pan-cancer AAC 0.32 5e-09
mRNA C1orf116 gCSI pan-cancer AAC 0.39 5e-09
mRNA B3GNT3 CCLE pan-cancer AAC 0.31 5e-09
mRNA GJB5 gCSI pan-cancer AAC 0.39 5e-09
mRNA LAMA5 gCSI pan-cancer AAC 0.41 5e-09
mRNA LSR CCLE pan-cancer AAC 0.34 5e-09
mRNA LAD1 CTRPv2 pan-cancer AAC 0.25 6e-09
mRNA CST6 CCLE pan-cancer AAC 0.29 6e-09
mRNA ALDH3A1 GDSC1000 pan-cancer AAC 0.3 7e-09
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