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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA SYT16 CCLE pan-cancer AAC 0.26 2e-08
mRNA ADGRF1 gCSI pan-cancer AAC 0.36 2e-08
mRNA CCT6A CTRPv2 pan-cancer AAC 0.19 2e-08
mRNA DSC2 CCLE pan-cancer AAC 0.29 2e-08
mRNA LCN2 gCSI pan-cancer AAC 0.35 2e-08
mRNA SCEL GDSC1000 pan-cancer AAC 0.27 2e-08
mRNA CLUL1 FIMM pan-cancer AAC 0.76 2e-08
mRNA KLK7 CCLE pan-cancer AAC 0.27 2e-08
mRNA PLEKHG6 CCLE pan-cancer AAC 0.29 2e-08
mRNA GRAMD2 CCLE pan-cancer AAC 0.26 2e-08
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