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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA TMEM125 CCLE pan-cancer AAC 0.33 2e-09
mRNA KLF5 gCSI pan-cancer AAC 0.45 2e-09
mRNA MKNK1 CTRPv2 pan-cancer AAC 0.21 2e-09
mRNA LYPD3 CCLE pan-cancer AAC 0.32 2e-09
mRNA EPS8L2 gCSI pan-cancer AAC 0.42 2e-09
mRNA CBLC CCLE pan-cancer AAC 0.32 2e-09
mRNA KLK5 CCLE pan-cancer AAC 0.29 2e-09
mRNA C1orf106 gCSI pan-cancer AAC 0.35 2e-09
mRNA MISP CCLE pan-cancer AAC 0.35 3e-09
mRNA CNKSR1 CCLE pan-cancer AAC 0.33 3e-09
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