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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA SEC61G CTRPv2 pan-cancer AAC 0.21 8e-10
mRNA LAMC2 gCSI pan-cancer AAC 0.41 8e-10
mRNA LIX1L CCLE pan-cancer AAC -0.32 9e-10
mRNA RBMS2 gCSI pan-cancer AAC 0.41 9e-10
mRNA PRSS8 GDSC1000 pan-cancer AAC 0.36 1e-09
mRNA FXYD3 CCLE pan-cancer AAC 0.33 1e-09
mRNA EPCAM CCLE pan-cancer AAC 0.39 1e-09
mRNA ITGB6 gCSI pan-cancer AAC 0.38 1e-09
mRNA ITGB4 CCLE pan-cancer AAC 0.34 1e-09
mRNA MPZL2 GDSC1000 pan-cancer AAC 0.34 1e-09
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