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Erlotinib

Synonyms

SourcesNames Used
CCLE, GDSC1000, GRAY, FIMM, UHNBreastErlotinib
gCSI, CTRPv2erlotinib
PharmacoGx Erlotinib

External IDs

DatabaseIdentifier
Smiles: COCCOC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)C#C)OCCOC.Cl
Inchikey: GTTBEUCJPZQMDZ-UHFFFAOYSA-N
Pubchem: 176871

Annotated Targets

EGFR, NR1I2, ERBB2

FDA Approval Status

Approved
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Top molecular features associated with response to Erlotinib


Feature TypeStandardized
Nominal ANOVA
mRNA KLK10 CCLE pan-cancer AAC 0.2 0.0002
mRNA DOK6 CTRPv2 pan-cancer AAC -0.13 0.0002
mRNA RGL3 CCLE pan-cancer AAC 0.19 0.0002
mRNA KRBOX4 CCLE pan-cancer AAC -0.17 0.0002
mRNA NFKBIZ GDSC1000 pan-cancer AAC 0.2 0.0002
mRNA MECOM gCSI pan-cancer AAC 0.24 0.0002
mRNA TMEM40 CCLE pan-cancer AAC 0.19 0.0002
mRNA DPYSL2 CTRPv2 pan-cancer AAC -0.14 0.0002
mRNA TTC21B gCSI pan-cancer AAC -0.22 0.0002
mRNA F3 CCLE pan-cancer AAC 0.22 0.0002
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