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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA EIF6 CTRPv2 pan-cancer AAC -0.078 0.03
mRNA PDIA4 CTRPv2 pan-cancer AAC -0.076 0.03
mRNA IRF2 CTRPv2 pan-cancer AAC -0.086 0.03
mRNA H2AFB1 CTRPv2 pan-cancer AAC -0.072 0.03
mRNA IRF9 CTRPv2 pan-cancer AAC -0.074 0.03
mRNA EIF4EBP1 CTRPv2 pan-cancer AAC 0.073 0.03
mRNA STK17B CTRPv2 pan-cancer AAC -0.085 0.03
mRNA ZNF317 CTRPv2 pan-cancer AAC 0.084 0.03
mRNA MRPL14 CTRPv2 pan-cancer AAC -0.073 0.03
mRNA HOXC9 CTRPv2 pan-cancer AAC 0.079 0.03
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