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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA PRSS57 CTRPv2 pan-cancer AAC 0.37 2e-28
mRNA GOLGA8M CTRPv2 pan-cancer AAC 0.33 2e-23
mRNA TIFAB CTRPv2 pan-cancer AAC 0.32 1e-22
mRNA DCANP1 CTRPv2 pan-cancer AAC 0.32 9e-22
mRNA ITGAL CTRPv2 pan-cancer AAC 0.35 3e-21
mRNA GOLGA8J CTRPv2 pan-cancer AAC 0.31 5e-20
mRNA GOLGA8T CTRPv2 pan-cancer AAC 0.26 2e-14
mRNA GOLGA8H CTRPv2 pan-cancer AAC 0.26 2e-14
mRNA GOLGA8N CTRPv2 pan-cancer AAC 0.27 2e-14
mRNA HMX3 CTRPv2 pan-cancer AAC 0.25 1e-13
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