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MGCD-265

Synonyms

SourcesNames Used
CTRPv2MGCD-265
PharmacoGx MGCD-265

External IDs

DatabaseIdentifier
Smiles: Cn1cnc(c1)-c1cc2nccc(Oc3ccc(NC(=S)NC(=O)Cc4ccccc4)cc3F)c2s1
Pubchem: 24901704

Annotated Targets

MET, TEK, MST1R, AXL, FLT1, FLT3, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to MGCD-265


Feature TypeStandardized
Nominal ANOVA
mRNA LIAS CTRPv2 pan-cancer AAC 0.076 0.04
mRNA CDK2AP2 CTRPv2 pan-cancer AAC -0.073 0.04
mRNA HNRNPL CTRPv2 pan-cancer AAC 0.074 0.04
mRNA ABHD17C CTRPv2 pan-cancer AAC -0.081 0.04
mRNA ARHGAP15 CTRPv2 pan-cancer AAC 0.095 0.04
mRNA HAUS1 CTRPv2 pan-cancer AAC 0.073 0.04
mRNA RPS5 CTRPv2 pan-cancer AAC 0.076 0.04
mRNA IMP4 CTRPv2 pan-cancer AAC -0.073 0.04
mRNA JTB CTRPv2 pan-cancer AAC -0.074 0.04
mRNA SLC22A18 CTRPv2 pan-cancer AAC -0.078 0.04
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