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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA SOCS2 GDSC1000 pan-cancer AAC 0.22 4e-12
mRNA GGT5 CTRPv2 pan-cancer AAC 0.24 6e-12
mRNA HBG2 GDSC1000 pan-cancer AAC 0.21 7e-12
mRNA SAMSN1 GDSC1000 pan-cancer AAC 0.31 9e-12
mRNA HSH2D CTRPv2 pan-cancer AAC 0.28 1e-11
mRNA FAM124B GDSC1000 pan-cancer AAC 0.22 2e-11
mRNA TAL1 GDSC1000 pan-cancer AAC 0.21 3e-11
mRNA TBXA2R GDSC1000 pan-cancer AAC 0.21 4e-11
mRNA ZNF175 GDSC1000 pan-cancer AAC 0.22 4e-11
mRNA LCP2 GDSC1000 pan-cancer AAC 0.29 5e-11
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