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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA LAPTM4B GDSC1000 pan-cancer AAC 0.34 4e-13
mRNA SIGLEC12 GDSC1000 pan-cancer AAC 0.24 5e-13
mRNA PRKCQ GDSC1000 pan-cancer AAC 0.24 6e-13
mRNA PTPN7 GDSC1000 pan-cancer AAC 0.38 6e-13
mRNA FAM117A CTRPv2 pan-cancer AAC 0.3 7e-13
mRNA ANK1 CTRPv2 pan-cancer AAC 0.25 8e-13
mRNA GATA1 GDSC1000 pan-cancer AAC 0.23 9e-13
mRNA C7orf34 CTRPv2 pan-cancer AAC 0.25 1e-12
mRNA LYL1 GDSC1000 pan-cancer AAC 0.32 1e-12
mRNA APOL4 GDSC1000 pan-cancer AAC 0.23 3e-12
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