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masitinib

Synonyms

SourcesNames Used
GDSC1000Masitinib
CTRPv2masitinib
PharmacoGx masitinib

External IDs

DatabaseIdentifier
Smiles: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
Pubchem: 10074640

Annotated Targets

KIT, FGFR3, PDGFRA, PDGFRB

FDA Approval Status

Not Approved
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Top molecular features associated with response to masitinib


Feature TypeStandardized
Nominal ANOVA
mRNA AC010287.1 CTRPv2 pan-cancer AAC 0.1 0.006
mRNA PLGLB2 GDSC1000 pan-cancer AAC 0.09 0.006
mRNA ZDHHC17 CTRPv2 pan-cancer AAC 0.1 0.006
mRNA CDKN3 GDSC1000 pan-cancer AAC -0.089 0.006
mRNA PCMT1 GDSC1000 pan-cancer AAC 0.088 0.006
mRNA CD2BP2 GDSC1000 pan-cancer AAC -0.086 0.006
mRNA DGCR8 CTRPv2 pan-cancer AAC 0.1 0.006
mRNA IL18BP GDSC1000 pan-cancer AAC 0.088 0.006
mRNA STXBP5 CTRPv2 pan-cancer AAC 0.099 0.006
mRNA CDC14A GDSC1000 pan-cancer AAC 0.095 0.006
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