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TKI258

Synonyms

SourcesNames Used
CCLETKI258
PharmacoGx TKI258

External IDs

DatabaseIdentifier
Smiles: CN1CCN(CC1)C2=CC3=C(C=C2)NC(=C4C(=C5C(=NC4=O)C=CC=C5F)N)N3
Inchikey: KCOYQXZDFIIGCY-ZZEZOPTASA-N
Pubchem: 9886808

FDA Approval Status

Not Approved
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Top molecular features associated with response to TKI258


Feature TypeStandardized
Nominal ANOVA
mRNA DCDC2B CCLE pan-cancer AAC -0.11 0.02
mRNA CD5L CCLE pan-cancer AAC -0.11 0.02
mRNA DMPK CCLE pan-cancer AAC -0.11 0.02
mRNA TRIM47 CCLE pan-cancer AAC -0.12 0.02
mRNA ZNF24 CCLE pan-cancer AAC 0.12 0.02
mRNA RPRD1B CCLE pan-cancer AAC -0.11 0.02
mRNA GALNT18 CCLE pan-cancer AAC -0.11 0.02
mRNA SAMD9 CCLE pan-cancer AAC -0.12 0.02
mRNA GATB CCLE pan-cancer AAC 0.11 0.02
mRNA PIK3C3 CCLE pan-cancer AAC 0.12 0.02
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