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GDC-0941

Synonyms

SourcesNames Used
GDSC1000GDC0941
gCSIgdc0941
FIMMPictilisib
CTRPv2GDC-0941
PharmacoGx GDC-0941

External IDs

DatabaseIdentifier
Smiles: CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6
Inchikey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
Pubchem: 17755052

Annotated Targets

PIK3CA, PIK3CB, PIK3CD, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to GDC-0941


Feature TypeStandardized
Nominal ANOVA
mRNA SYT4 gCSI pan-cancer AAC -0.19 0.006
mRNA KIF19 gCSI pan-cancer AAC -0.17 0.006
mRNA VIL1 gCSI pan-cancer AAC -0.2 0.006
mRNA GPR3 gCSI pan-cancer AAC -0.18 0.006
mRNA DTX4 gCSI pan-cancer AAC 0.18 0.006
mRNA MAN2A2 gCSI pan-cancer AAC -0.17 0.006
mRNA BTG2 gCSI pan-cancer AAC 0.2 0.006
mRNA MYBL1 gCSI pan-cancer AAC 0.17 0.005
mRNA MIER3 gCSI pan-cancer AAC 0.16 0.005
mRNA CDIP1 gCSI pan-cancer AAC -0.17 0.005
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