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GDC-0941

Synonyms

SourcesNames Used
GDSC1000GDC0941
gCSIgdc0941
FIMMPictilisib
CTRPv2GDC-0941
PharmacoGx GDC-0941

External IDs

DatabaseIdentifier
Smiles: CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6
Inchikey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
Pubchem: 17755052

Annotated Targets

PIK3CA, PIK3CB, PIK3CD, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to GDC-0941


Feature TypeStandardized
Nominal ANOVA
mRNA ADGRF3 GDSC1000 pan-cancer AAC 0.1 0.003
mRNA ADORA2B CTRPv2 pan-cancer AAC -0.15 9e-05
mRNA ADRB2 gCSI pan-cancer AAC 0.18 0.006
mRNA AFMID CTRPv2 pan-cancer AAC 0.12 0.002
mRNA AGA gCSI pan-cancer AAC 0.17 0.006
mRNA AGAP3 gCSI pan-cancer AAC -0.2 0.002
mRNA AGPAT1 CTRPv2 pan-cancer AAC -0.13 0.002
mRNA AHCYL2 CTRPv2 pan-cancer AAC 0.1 0.005
mRNA AHI1 gCSI pan-cancer AAC -0.16 0.006
mRNA AICDA gCSI pan-cancer AAC 0.24 0.0002
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