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GDC-0941

Synonyms

SourcesNames Used
GDSC1000GDC0941
gCSIgdc0941
FIMMPictilisib
CTRPv2GDC-0941
PharmacoGx GDC-0941

External IDs

DatabaseIdentifier
Smiles: CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6
Inchikey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
Pubchem: 17755052

Annotated Targets

PIK3CA, PIK3CB, PIK3CD, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to GDC-0941


Feature TypeStandardized
Nominal ANOVA
mRNA ACTN4 CTRPv2 pan-cancer AAC -0.11 0.005
mRNA ACTR10 gCSI pan-cancer AAC 0.17 0.004
mRNA ACVR2B gCSI pan-cancer AAC -0.18 0.003
mRNA ACYP1 FIMM pan-cancer AAC -0.62 0.0005
mRNA ADAMTSL3 gCSI pan-cancer AAC 0.2 0.003
mRNA ADAP2 gCSI pan-cancer AAC 0.21 0.001
mRNA ADAR CTRPv2 pan-cancer AAC 0.13 0.0003
mRNA ADCY1 GDSC1000 pan-cancer AAC -0.15 8e-05
mRNA ADCY6 FIMM pan-cancer AAC 0.62 0.003
mRNA ADCYAP1 gCSI pan-cancer AAC -0.18 0.004
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