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GDC-0941

Synonyms

SourcesNames Used
GDSC1000GDC0941
gCSIgdc0941
FIMMPictilisib
CTRPv2GDC-0941
PharmacoGx GDC-0941

External IDs

DatabaseIdentifier
Smiles: CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6
Inchikey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
Pubchem: 17755052

Annotated Targets

PIK3CA, PIK3CB, PIK3CD, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to GDC-0941


Feature TypeStandardized
Nominal ANOVA
mRNA PRLH FIMM pan-cancer AAC -0.53 0.002
mRNA PORCN FIMM pan-cancer AAC -0.52 0.002
mRNA NELFE FIMM pan-cancer AAC -0.52 0.003
mRNA PBOV1 FIMM pan-cancer AAC -0.51 0.005
mRNA ICAM1 FIMM pan-cancer AAC -0.51 0.003
mRNA STS FIMM pan-cancer AAC -0.51 0.002
mRNA PGM1 FIMM pan-cancer AAC -0.5 0.005
mRNA SLC30A1 FIMM pan-cancer AAC -0.49 0.003
mRNA KYAT1 FIMM pan-cancer AAC -0.48 0.006
mRNA RGL1 FIMM pan-cancer AAC -0.48 0.005
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