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GDC-0941

Synonyms

SourcesNames Used
GDSC1000GDC0941
gCSIgdc0941
FIMMPictilisib
CTRPv2GDC-0941
PharmacoGx GDC-0941

External IDs

DatabaseIdentifier
Smiles: CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6
Inchikey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
Pubchem: 17755052

Annotated Targets

PIK3CA, PIK3CB, PIK3CD, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to GDC-0941


Feature TypeStandardized
Nominal ANOVA
mRNA KCNK6 CTRPv2 pan-cancer AAC -0.1 0.005
mRNA TSPAN14 GDSC1000 pan-cancer AAC 0.098 0.005
mRNA STPG1 GDSC1000 pan-cancer AAC -0.091 0.005
mRNA MYBL1 gCSI pan-cancer AAC 0.17 0.005
mRNA PDLIM1 GDSC1000 pan-cancer AAC 0.1 0.006
mRNA FER CTRPv2 pan-cancer AAC -0.1 0.006
mRNA KBTBD8 GDSC1000 pan-cancer AAC 0.12 0.006
mRNA PTPN11 FIMM pan-cancer AAC 0.49 0.006
mRNA MEX3C CTRPv2 pan-cancer AAC 0.11 0.006
mRNA MBD1 CTRPv2 pan-cancer AAC 0.11 0.006
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