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GDC-0941

Synonyms

SourcesNames Used
GDSC1000GDC0941
gCSIgdc0941
FIMMPictilisib
CTRPv2GDC-0941
PharmacoGx GDC-0941

External IDs

DatabaseIdentifier
Smiles: CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6
Inchikey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
Pubchem: 17755052

Annotated Targets

PIK3CA, PIK3CB, PIK3CD, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to GDC-0941


Feature TypeStandardized
Nominal ANOVA
mRNA ST18 GDSC1000 pan-cancer AAC -0.13 0.0001
mRNA USP7 CTRPv2 pan-cancer AAC 0.15 0.0001
mRNA PIP4K2C GDSC1000 pan-cancer AAC -0.15 0.0001
mRNA LIN28B GDSC1000 pan-cancer AAC -0.14 0.0001
mRNA GRAP2 CTRPv2 pan-cancer AAC -0.14 0.0001
mRNA UCK2 gCSI pan-cancer AAC -0.22 0.0001
mRNA CNKSR3 gCSI pan-cancer AAC -0.28 0.0001
mRNA MFN2 GDSC1000 pan-cancer AAC -0.13 0.0001
mRNA MGEA5 gCSI pan-cancer AAC 0.23 0.0001
mRNA UBAP2 CTRPv2 pan-cancer AAC 0.15 0.0001
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