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GDC-0941

Synonyms

SourcesNames Used
GDSC1000GDC0941
gCSIgdc0941
FIMMPictilisib
CTRPv2GDC-0941
PharmacoGx GDC-0941

External IDs

DatabaseIdentifier
Smiles: CS(=O)(=O)N1CCN(CC1)CC2=CC3=C(S2)C(=NC(=N3)C4=C5C=NNC5=CC=C4)N6CCOCC6
Inchikey: LHNIIDJUOCFXAP-UHFFFAOYSA-N
Pubchem: 17755052

Annotated Targets

PIK3CA, PIK3CB, PIK3CD, PIK3CG

FDA Approval Status

Not Approved
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Top molecular features associated with response to GDC-0941


Feature TypeStandardized
Nominal ANOVA
mRNA PHF1 CTRPv2 pan-cancer AAC -0.15 5e-05
mRNA GAMT CTRPv2 pan-cancer AAC 0.15 6e-05
mRNA CYB561A3 CTRPv2 pan-cancer AAC 0.15 6e-05
mRNA DLL4 gCSI pan-cancer AAC -0.25 6e-05
mRNA CHCHD6 GDSC1000 pan-cancer AAC -0.15 6e-05
mRNA RIMKLA GDSC1000 pan-cancer AAC -0.14 6e-05
mRNA DBNDD2 CTRPv2 pan-cancer AAC -0.16 7e-05
mRNA CIC CTRPv2 pan-cancer AAC 0.15 7e-05
mRNA ZNF175 gCSI pan-cancer AAC -0.23 7e-05
mRNA E2F5 CTRPv2 pan-cancer AAC 0.15 7e-05
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