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PLX4720

Synonyms

SourcesNames Used
CCLE, GDSC1000PLX4720
CTRPv2PLX-4720
PharmacoGx PLX4720

External IDs

DatabaseIdentifier
Smiles: CCCS(=O)(=O)NC1=C(C(=C(C=C1)F)C(=O)C2=CNC3=NC=C(C=C23)Cl)F
Inchikey: YZDJQTHVDDOVHR-UHFFFAOYSA-N
Pubchem: 24180719

Annotated Targets

BRAF, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to PLX4720


Feature TypeStandardized
Nominal ANOVA
mRNA SLC45A2 CCLE pan-cancer AAC 0.35 9e-12
mRNA SHC4 CCLE pan-cancer AAC 0.39 2e-11
mRNA TLR8 CCLE pan-cancer AAC 0.27 1e-10
mRNA FMN1 CCLE pan-cancer AAC 0.3 1e-10
mRNA TYR CCLE pan-cancer AAC 0.36 2e-10
mRNA PLA1A CCLE pan-cancer AAC 0.31 4e-10
mRNA MMP8 CCLE pan-cancer AAC 0.4 5e-10
mRNA SOX10 CCLE pan-cancer AAC 0.45 1e-09
mRNA PMEL CCLE pan-cancer AAC 0.31 2e-09
mRNA LRRK2 CCLE pan-cancer AAC 0.3 2e-09
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