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PLX4720

Synonyms

SourcesNames Used
CCLE, GDSC1000PLX4720
CTRPv2PLX-4720
PharmacoGx PLX4720

External IDs

DatabaseIdentifier
Smiles: CCCS(=O)(=O)NC1=C(C(=C(C=C1)F)C(=O)C2=CNC3=NC=C(C=C23)Cl)F
Inchikey: YZDJQTHVDDOVHR-UHFFFAOYSA-N
Pubchem: 24180719

Annotated Targets

BRAF, KDR

FDA Approval Status

Not Approved
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Top molecular features associated with response to PLX4720


Feature TypeStandardized
Nominal ANOVA
mRNA PLP1 GDSC1000 pan-cancer AAC 0.36 2e-14
mRNA SDC3 CTRPv2 pan-cancer AAC 0.37 3e-15
mRNA GAPDHS CCLE pan-cancer AAC 0.37 3e-17
mRNA NFATC2 CTRPv2 pan-cancer AAC 0.37 3e-19
mRNA MIA-RAB4B CTRPv2 pan-cancer AAC 0.37 8e-20
mRNA MLANA CCLE pan-cancer AAC 0.38 3e-12
mRNA RXRG CTRPv2 pan-cancer AAC 0.38 6e-22
mRNA SHC4 CCLE pan-cancer AAC 0.39 2e-11
mRNA MMP8 CCLE pan-cancer AAC 0.4 5e-10
mRNA CPN1 CCLE pan-cancer AAC 0.4 3e-12
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