1. Home/
  2. Compounds/
  3. BX-912

BX-912

Synonyms

SourcesNames Used
GDSC1000BX-912
PharmacoGx BX-912

External IDs

DatabaseIdentifier
Smiles: Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc4c[nH]cn4
Pubchem: 11754511

Annotated Targets

CDK2, CHEK1, GSK3B, KDR, PDK1, PDPK1

FDA Approval Status

Not Approved
Dataset Select
Download Data as CSV

Top molecular features associated with response to BX-912


Feature TypeStandardized
Nominal ANOVA
mRNA TNRC6C GDSC1000 pan-cancer AAC 0.25 4e-15
mRNA MDFI GDSC1000 pan-cancer AAC 0.25 6e-15
mRNA GALE GDSC1000 pan-cancer AAC -0.26 9e-15
mRNA ATOX1 GDSC1000 pan-cancer AAC -0.25 1e-14
mRNA PRPF4B GDSC1000 pan-cancer AAC 0.24 1e-14
mRNA TTF1 GDSC1000 pan-cancer AAC 0.24 1e-14
mRNA SHPRH GDSC1000 pan-cancer AAC 0.25 2e-14
mRNA TMEM170B GDSC1000 pan-cancer AAC 0.25 2e-14
mRNA ABHD17B GDSC1000 pan-cancer AAC 0.24 2e-14
mRNA ZNF627 GDSC1000 pan-cancer AAC 0.23 2e-14
Download CSV