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BX-912

Synonyms

SourcesNames Used
GDSC1000BX-912
PharmacoGx BX-912

External IDs

DatabaseIdentifier
Smiles: Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc4c[nH]cn4
Pubchem: 11754511

Annotated Targets

CDK2, CHEK1, GSK3B, KDR, PDK1, PDPK1

FDA Approval Status

Not Approved
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Top molecular features associated with response to BX-912


Feature TypeStandardized
Nominal ANOVA
mRNA KIAA1143 GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA HSPG2 GDSC1000 pan-cancer AAC -0.12 0.0002
mRNA ZBTB40 GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA SH2D3A GDSC1000 pan-cancer AAC -0.14 0.0002
mRNA RCOR3 GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA CNOT9 GDSC1000 pan-cancer AAC 0.12 0.0002
mRNA CCR2 GDSC1000 pan-cancer AAC 0.11 0.0002
mRNA STYXL1 GDSC1000 pan-cancer AAC -0.11 0.0002
mRNA CSRNP1 GDSC1000 pan-cancer AAC -0.11 0.0002
mRNA ITK GDSC1000 pan-cancer AAC 0.12 0.0002
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