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BX-912

Synonyms

SourcesNames Used
GDSC1000BX-912
PharmacoGx BX-912

External IDs

DatabaseIdentifier
Smiles: Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc4c[nH]cn4
Pubchem: 11754511

Annotated Targets

CDK2, CHEK1, GSK3B, KDR, PDK1, PDPK1

FDA Approval Status

Not Approved
Dataset Select
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Top molecular features associated with response to BX-912


Feature TypeStandardized
Nominal ANOVA
mRNA MEX3A GDSC1000 pan-cancer AAC 0.28 2e-16
mRNA CAST GDSC1000 pan-cancer AAC -0.28 2e-16
mRNA MSL2 GDSC1000 pan-cancer AAC 0.3 2e-16
mRNA PDS5B GDSC1000 pan-cancer AAC 0.27 3e-16
mRNA BCL11A GDSC1000 pan-cancer AAC 0.27 3e-16
mRNA BAHCC1 GDSC1000 pan-cancer AAC 0.24 4e-16
mRNA TMBIM1 GDSC1000 pan-cancer AAC -0.28 8e-16
mRNA BCL11B GDSC1000 pan-cancer AAC 0.25 1e-15
mRNA ZBTB38 GDSC1000 pan-cancer AAC -0.24 1e-15
mRNA ZNF445 GDSC1000 pan-cancer AAC 0.27 3e-15
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