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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA A2M GDSC1000 pan-cancer AAC 0.18 6e-08
mRNA AARS2 CTRPv2 pan-cancer AAC 0.17 0.0007
mRNA AASS GDSC1000 pan-cancer AAC 0.19 8e-09
mRNA AATF CTRPv2 pan-cancer AAC 0.25 5e-08
mRNA AATK-AS1 CTRPv2 pan-cancer AAC 0.18 0.0004
mRNA ABCA9 CTRPv2 pan-cancer AAC 0.18 9e-05
mRNA ABCB4 CTRPv2 pan-cancer AAC 0.17 0.0003
mRNA ABCD1 CTRPv2 pan-cancer AAC 0.22 6e-06
mRNA ABCF1 GDSC1000 pan-cancer AAC -0.13 1e-05
mRNA ABCG5 CTRPv2 pan-cancer AAC 0.24 3e-07
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