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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA IKZF1 GDSC1000 pan-cancer AAC -0.32 9e-06
mRNA ARHGAP30 GDSC1000 pan-cancer AAC -0.32 3e-06
mRNA CORO1A GDSC1000 pan-cancer AAC -0.25 1e-05
mRNA VASN CTRPv2 pan-cancer AAC -0.21 7e-05
mRNA PODN CTRPv2 pan-cancer AAC -0.21 2e-05
mRNA MSL2 GDSC1000 pan-cancer AAC -0.2 4e-08
mRNA PPP4R3A GDSC1000 pan-cancer AAC -0.19 1e-08
mRNA CD248 CTRPv2 pan-cancer AAC -0.19 0.0001
mRNA ADCY4 CTRPv2 pan-cancer AAC -0.19 4e-05
mRNA PCDH18 CTRPv2 pan-cancer AAC -0.19 9e-05
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