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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA JAG2 GDSC1000 pan-cancer AAC -0.19 9e-08
mRNA C1QTNF5 CTRPv2 pan-cancer AAC -0.19 0.0002
mRNA MFRP CTRPv2 pan-cancer AAC -0.19 0.0002
mRNA VCPKMT GDSC1000 pan-cancer AAC -0.19 4e-09
mRNA KRTAP1-5 CTRPv2 pan-cancer AAC -0.19 0.0001
mRNA C16orf87 GDSC1000 pan-cancer AAC -0.18 3e-08
mRNA NKAPL CTRPv2 pan-cancer AAC -0.18 9e-05
mRNA LLGL2 GDSC1000 pan-cancer AAC -0.18 7e-06
mRNA GREM1 CTRPv2 pan-cancer AAC -0.18 0.0001
mRNA DCN CTRPv2 pan-cancer AAC -0.18 0.0001
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