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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA INA GDSC1000 pan-cancer AAC -0.11 0.0009
mRNA FOXN1 GDSC1000 pan-cancer AAC -0.099 0.0009
mRNA SPEN GDSC1000 pan-cancer AAC -0.11 0.0009
mRNA C5AR1 GDSC1000 pan-cancer AAC -0.1 0.0009
mRNA KCNQ2 GDSC1000 pan-cancer AAC -0.1 0.0009
mRNA SMAD9 GDSC1000 pan-cancer AAC -0.11 0.0009
mRNA TSPO GDSC1000 pan-cancer AAC 0.11 0.0009
mRNA MED15 GDSC1000 pan-cancer AAC 0.1 0.0009
mRNA INHBB GDSC1000 pan-cancer AAC -0.11 0.0009
mRNA MED30 GDSC1000 pan-cancer AAC -0.11 0.0009
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