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dabrafenib

Synonyms

SourcesNames Used
GDSC1000Dabrafenib
CTRPv2dabrafenib
PharmacoGx dabrafenib

External IDs

DatabaseIdentifier
Smiles: CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2c(F)cccc2F)c1F
Pubchem: 44462760

Annotated Targets

BRAF, LIMK1, NEK11, RAF1, SIK1

FDA Approval Status

Approved
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Top molecular features associated with response to dabrafenib


Feature TypeStandardized
Nominal ANOVA
mRNA FOXO3 GDSC1000 pan-cancer AAC -0.12 6e-05
mRNA ACO1 GDSC1000 pan-cancer AAC 0.13 6e-05
mRNA SFXN3 CTRPv2 pan-cancer AAC 0.21 6e-05
mRNA SLC2A8 GDSC1000 pan-cancer AAC -0.13 6e-05
mRNA ITGB1 GDSC1000 pan-cancer AAC 0.15 7e-05
mRNA CEMP1 CTRPv2 pan-cancer AAC 0.19 7e-05
mRNA CORO2B CTRPv2 pan-cancer AAC 0.19 7e-05
mRNA STEAP1B GDSC1000 pan-cancer AAC 0.13 7e-05
mRNA IER3 GDSC1000 pan-cancer AAC 0.15 7e-05
mRNA GPR143 GDSC1000 pan-cancer AAC 0.13 7e-05
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